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VU0810464

Glpbio
Catalog No:GC39459-10mM (in 1mL DMSO) CAS No.:2126040-21-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:VU0810464 是有效的,选择性的非尿素蛋白门控的内向整流钾通道 (GIRK, Kir3) 激活剂。 VU0810464 对神经元 GIRK1/2 (EC50=165 nM) 和 GIRK1/4 (EC50=720 nM) 神经通道具有纳摩尔效价,并且具有脑部渗透性。DMSO: ≥ 250 mg/mL (714.63 mM)
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